Abstract:Objective: To study the chemical constituents of the Tibetan medicine Caryopteris toroetii. Method: The crude drug was extracted with 95% EtOH and isolated by repeatedly chromatographic methods. The structures of the isolated compounds were elucidated by spectral analysis. Result: Six compounds were yielded and identified as: phenethyl cinnamide (1), 1 hydroxy 2, 3, 4, 5 tetramethoxy xanthone (2), 1 hydroxy 2, 3, 5 trimethoxy xanthone (3), (2S) 5 hydroxy 7 methoxyflavanone (4), 2′, 4′ dihydroxydihydrochalcone (5) and rutin (6). Conclusion: All the above compounds were obtained from C. toroetii for the first time.